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Found 4 results
Filtros: Palavra-chave is Antimalarials  [Clear All Filters]
2015
Horta P, Kuş N, Henriques MSofia C, et al. Quinolone-Hydroxyquinoline Tautomerism in Quinolone 3-Esters. Preserving the 4-Oxoquinoline Structure To Retain Antimalarial Activity. J Org Chem. 2015;80(24):12244-57. doi:10.1021/acs.joc.5b02169
2010
Gibbons P, Verissimo E, Araujo NC, et al. Endoperoxide carbonyl falcipain 2/3 inhibitor hybrids: toward combination chemotherapy of malaria through a single chemical entity. J Med Chem. 2010;53(22):8202-6. doi:10.1021/jm1009567
2009
Araújo NCP, Barton V, Jones M, et al. Semi-synthetic and synthetic 1,2,4-trioxaquines and 1,2,4-trioxolaquines: synthesis, preliminary SAR and comparison with acridine endoperoxide conjugates. Bioorg Med Chem Lett. 2009;19(7):2038-43. doi:10.1016/j.bmcl.2009.02.013
2008
Verissimo E, Berry N, Gibbons P, et al. Design and synthesis of novel 2-pyridone peptidomimetic falcipain 2/3 inhibitors. Bioorg Med Chem Lett. 2008;18(14):4210-4. doi:10.1016/j.bmcl.2008.05.068